【药物名称】Meloxicam, UH-AC 62XX, Mobicox, Movatec, Tenaron, Parocin, Movalis, Mobec, Mobic, Metacam
化学结构式(Chemical Structure):
参考文献No.109638
标题:MELOXICAM < Rec INN >
作者:Trummlitz, G.; Engelhardt, G.; Busch, U.
来源:Drugs Fut 1989,14(11),1047
合成路线图解说明:

The synthesis of meloxicam is performed as follows: The reaction of benzisothiazolo-3(2H)-one-1,1-dioxide (I) with methyl chloroacetate gives the methyl 2(3H)-acetate derivative, which is isomerized with sodium methoxide in toluene/tert-butanol yielding methyl 4-hydroxy-2H-1,2-benzothiazine-3-carboxylate-1,1-dioxide. The subsequent methylation with methyl iodide in methanol yields 2-methyl compound (II). Finally, this compound is treated with 2-amino-5-methylthiazole in xylene.

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