【药物名称】XR-3054
化学结构式(Chemical Structure):
参考文献No.543945
标题:XR 3054, structurally related to limonene, is a novel inhibitor of farnesyl protein transferase
作者:Donaldson, M.J.; Skoumas, V.; Watson, M.; Ashworth, P.A.; Ryder, H.; Moore, M.; Coombes, R.C.
来源:Eur J Cancer 1999,35(6),1014
合成路线图解说明:

Sharpless asymmetric epoxidation of (S)-(-)-perillyl alcohol (I) using tert-butyl hydroperoxide and diethyl L-tartrate produced epoxide (II), which was reduced to diol (III) by means of LiAlH4 in cold THF. Treatment of (III) with 2,2-dimethoxypropane (IV) and p-toluenesulfonic acid then furnished the title isopropylidene ketal.

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