【药物名称】GT-3381, CHF-3381
化学结构式(Chemical Structure):
参考文献No.35632
标题:alpha-Amino acid amides, preparation thereof and the therapeutical use thereof
作者:Chiesi, P.; Ventura, P.; Delcanale, M.; De Fanti, R.; Armani, E.; Villetti, G.; Pietra, C. (Chiesi Farmaceutici SpA)
来源:EP 0951465; JP 2001506577; US 6114391; WO 9803472
合成路线图解说明:

The reductive condensation between 2-indanone (I) and glycine methyl ester (II) in the presence of sodium cyanoborohydride furnished methyl (2-indanylamino)acetate (III). Subsequent ammonolysis of the methyl ester group of (III) in methanolic ammonia gave the glycinamide derivative (IV), which was finally converted to the title hydrochloride salt.

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