【药物名称】ProVP-16II
化学结构式(Chemical Structure):
参考文献No.666184
标题:Synthesis, hydrolytic activation and cytotoxicity of etoposide prodrugs
作者:Wrasidlo, W.; Schroder, U.; Bernt, K.; Hubener, N.; Shabat, D.; Gaedicke, G.; Lode, H.
来源:Bioorg Med Chem Lett 2002,12(4),557
合成路线图解说明:

Condensation of etoposide (I) with 2,2-dimethyl-1,3-dioxolan-4-ylmethyl chloroformate (II) provides the carbonate ester (III). Then, acidic hydrolysis of the acetonide group of (III) leads to the target compound.

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