【药物名称】
化学结构式(Chemical Structure):
参考文献No.761554
标题:Arachidonylsulfonyl derivatives as cannabinoid CB1 receptor and fatty acid amide hydrolase inhibitors
作者:Segall, Y.; Quistad, G.B.; Nomura, D.K.; Casida, J.E.
来源:Bioorg Med Chem Lett 2003,13(19),3301
合成路线图解说明:

Arachidonic acid (I) is reduced with LiAlH4 to the primary alcohol (II), which is subsequently brominated to (III) upon treatment with CBr4 and PPh3. After conversion of bromide (III) into the corresponding Grignard reagent, reaction with sulfuryl chloride furnishes the sulfononic acid chloride (IV). Finally, chloride (IV) is converted into the title sulfonyl fluoride by displacement with tetrabutylammonium fluoride in THF.

Drug Information Express,Drug R&D,Chemical Database,Patent Search.
Copyright © 2006-2024 Drug Future. All rights reserved.Contact Us